Angiogenesis, Inflammation & Therapeutics | Online ISSN  2207-872X
RESEARCH ARTICLE   (Open Access)

In Vitro Anti-Inflammatory Potential of Mangifera Indica Peels

Bhaskaran Sathyapriya1, Jayesh S Raghavendra2, Swamikannu Bhuminathan3, Adugula Chandrakala4, Kesavaram Padmavathy5*, Bharathwaj D K6, Indhumathi Krishnaswamy6

+ Author Affiliations

Journal of Angiotherapy 5 (2) 1-5 https://doi.org/10.25163/angiotherapy.521214422315151221

Submitted: 23 November 2021 Revised: 26 November 2021  Published: 15 December 2021 


Abstract

Background: Mangifera indica including the peels, are valued for their therapeutic applications, including anti-inflammatory effects. Previous studies have highlighted the rich bioactive profile of Mangifera indica, including polyphenols, flavonoids, and tannins, which contribute to its diverse pharmacological activities. Methods: Fresh mango peels were collected, dried, and powdered. The peel powder was extracted using 80% acetone, and the extract was concentrated and stored for analysis. The anti-inflammatory activity was assessed via a protein denaturation inhibition assay, involving a reaction mixture of bovine serum albumin (BSA) with varying concentrations of the peel extract. The assay measured the extent of protein denaturation induced by heat, with the percentage inhibition calculated spectrophotometrically at 660 nm. Aspirin was used as a standard for comparison. Results: Mangifera indica peel extracts exhibited significant anti-inflammatory activity, with inhibition of protein denaturation increasing in a dose-dependent manner. At a concentration of 500 µg/mL, the extract achieved a maximum inhibition of 71.93 ± 1.12%. The IC50 value was determined to be 119.35 ± 1.99 µg/mL. Aspirin, at 200 µg/mL, showed a maximum inhibition of 77.12 ± 1.42%. These results suggest that the anti-inflammatory efficacy of Mangifera indica peel extracts is comparable to that of aspirin. Conclusion: This study demonstrates that Mangifera indica peels possess significant anti-inflammatory activity, attributed to their polyphenol content and ability to inhibit protein denaturation.

Keywords: Mangifera indica, Anti-inflammatory, Protein denaturation, Peel extracts, Bioactive compounds

Introduction

GO

Mangifera indica (MI) has been an important herb in the Ayurveda and native medicine for more than four thousand years. Mangoes lie in the genus Mangifera consisting of over thirty taxonomic tropic fruit trees in the plant family Anacardiaceae.

Different parts of MI exhibits multi - medicinal properties as per Ayurvedic medicine(Scartezzini P, Speroni E 2000). It is a polyphenolic antioxidant with anti lipid peroxidation, immunomodulator, hypotensive and antidiabetic properties.

Several components of MI are utilized as a disinfectant, hemostatic, sudorific, anthelmintic, purgative and also used in the medical management of  looseness of the bowels, infectious disease, blood disorder, respiratory illness,  high blood pressure, sleep disorder, autoimmune disease, odontalgia, bleeding and hemorrhoids.( Khan MN et al., 2000). It is also used in the treatment of abscesses, animal bite, neoplasm, toxic condition, spontaneous abortion, zoonotic disease, vesicle and hepatic disease disorders.( Khan MN et al., a 1993).

The seed kernel of MI exhibits evidential anti-inflammatory property in acute and chronic inflammation.(Shankarnarayanan D et al., 1979 Khan MA, Khan MN b 1989). The leaf extract of MI also displays antibacterial and analgesic properties. (Ross 1999). All the properties were found due to the presence of polyphenols in the extract. Anti-inflammatory property of MI extracts were studied by topical injection of  0.5-2 mg of MI extract in the ear of mice.( Subbarayan C, Cama HR 1966, Seifried HE et al., 2007).  The topical administration of MI extract decreased ear swelling evoked by arachidonic acid and phorbol myristate in rat. (Diplock AT et al.,1998, Maxwell SR 1997). The anti-inflammatory and anti-nociceptive activities of MI extract are evident from the study results conducted on rat.( Martinez G et al.,2007, Pardo-Andreu GL et al., 2006, Rocha Ribeiro SM et al., 2007).

MI is a giant coniferous woody plant in the Anacardiaceae family with a height of about 46 meters,  concave-shaped and heavily bifurcate from a sturdy tree trunk. The leaf blades are almost 26-cm long and 8-cm broader, and spirally arranged leaves produce an aroma when crushed. There are about  4000 tiny  yellowish-green flowers. When ripened, the fruit shows a greater variation in form and size with a  yellow pulp, solitary seed, and yellowish red skin. The various chemical substance of MI includes the polyphenols, flavonoids, gallic acid, tannins &  derivatives.

Antioxidant and antiproliferative activity

The oxidative impairment evoked by hydrogen peroxide in a human hepatoma cell, HepG2 were reversed by the cytoprotective phenomenon of mango pulp and skin extracts and the fundamental chemical process was determined by a single-cell electrophoresis assay. DNA damage was inhibited by the management of HepG2 cell with MI skin extract. Eectron spin resonance (ESR) was used to evaluate the free radical scavenging properties of MI pulp and skin extracts. The mango skin possesses powerful free radical scavenging quality on diphenyl picrylhydrazyl and alkyl radicals than mango pulp, irrespective of maturity.( Shibahara A,et al.,1993, Nunez Selles AJ et al.,2002, Andreas Set al.,2007).  Skin extract displayed a significant antiproliferative effect against cancer cells than flesh extract attributed to phenolic and flavonoid.( Pott Iet al., 2003). The results showed the skin extract poetesses great antioxidant activity and anticancer properties.( Chen JP et al., 2004).

Mango, an important tropical fruits is processed for various products during which the skin is often being wasted. The bioactive conserves extracted from raw and ripe mango skin using 80% acetone were subjected to acid hydrolysis. Gallic acid, syringic acid, mangiferin, ellagic acid, gentisyl-protocatechuic acid, quercetin were the phenolic compounds identified in both raw and ripe peels. In addition to this, glycosylated iriflophenone and maclurin derivatives were also seen in raw peel. ß-Carotene and lutein were the major carotenoids. Thus, raw and ripe mango peel extracts have different phenolic compounds and carotenoids with various pharmaceutical applications.

Polyphenoloxidase from MI skin was refined to homogeneity by ammonium sulphate fractionation, chromatography on DEAE-Sephadex and gel filtration of Sephadex G-200. The enzyme had an apparent molecular weight of 136,000. Its pH and temperature optimum were 5.4 and 50‡C, respectively. Mango skin polyphenol oxidase, when immobilized onto DEAE Sephadex showed slightly higher Km for catechol and lower pH and temperature optima.

Materials and Method

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protein denaturation inhibition assay. Inflammation is caused by protein denaturation and therefore it can be used for in vitro screening. Test extract at various concentrations with 1% aqueous solution of bovine albumin is the reaction mixture, the pH adjusted using 1N hydrochloric acid. 

The samples were incubated at 37oC for 20 min and heated at  57oC for  20  min. The turbidity was measured spectrophotometrically at 660nm after cooling the samples..[10, 11]

Percentage inhibition  of  protein  denaturation was determined using the formula: 

Percentage  inhibition  =  (Abs control  –  Abs sample) X 100/ Abs control

Results

GO

The documented reason of inflammation is protein denaturation. As a part of the research on the mechanism of anti-inflammatory property, the quality of the extract to inhibit protein denaturation was also investigated. It was efficient in decreasing heat-induced albumin denaturation at various concentrations, as shown in table 1 Maximum inhibition 71.93±1.117% was observed at 500µg/ml. IC50 value was found to be  119.35±1.99µg/ml  Aspirin, a  standard anti-inflammatory drug showed the maximum inhibition, 77.12±1.42% at the  concentration of  200µg/ml (Table 1).  

Table 1. Protein denaturation Inhibiting activity of the methanolic extract

Sample concentration (µg)

Percentage activity

%

Control

(Aspirin) Concentration(µg)

 

Percentage activity

%

 

100

7.42 ± 0.89

50

17.97±0.50

200

19.23 ± 1.79

100

32.68±0.57

300

35.25 ± 1.22

150

47.39±1.50

400

52.53 ± 1.22

200

63.07±1.49

500

72.93 ± 1.117

250

77.12±1.42

Ic 50 ( µg/ml)

102.35±1.99

Ic 50 ( µg/ml)

39.78±0.50

 

Discussion

GO

The seed kernel of MI exhibits evidentiary anti-inflammatory activity in acute and chronic inflammation. (Muruganandan S et al.,2003, Desai PDet al.,1996) The leaf extract of MI also displays antibacterial and analgesic properties. All the properties were found due to the presence of polyphenols in the extract. Mangifera indica is an essential source of many pharmacologically and medicinally important chemicals such as mangiferin, polyphenols and carotenes. (Knödler Met al., 2007, Ornelas-Paz Jde J et al., 2007, Subha R et al.,2007). Many different pharmacological activities, antioxidant, radioprotective, immunomodulatory, anti-allergic, antidiabetic, lipolytic, monoamine oxidase-inhibiting and antimicrobial have been reported for mangiferin.  A defined mixture of components like polyphenols, terpenoids, steroids, fatty acids, and microelements is present in VIMANG, an extract from the stem bark of M. indica. In order to study whether the extract contributes to this mechanism of anti-inflammatory activity, inhibitory effects of M. indica are bestowed in this work on in vitro eicosanoid-releasing systems. ( Gabino G et al., 2008, Pardo Andreu Get al.,2005, Sanchez GMet al.,2000).

Conclusion

GO

This study reveals that Mangnifera indica has varied pharmacological activities and alsoan essential source of pharmacologically and medicinally powerful chemicals such as mangiferin, polyphenols and carotenes. Due to its various activities and therapeutic use.of mangiferin, it has been used with success in Ayurveda for many years .

Author contribution

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Bhaskaran Sathyapriya conceived of the presented idea. Jayesh S Raghavendra, Swamikannu Bhuminathan  Adugula Chandrakala, Kesavaram Padmavathy, Bharathwaj D K and Indhumathi Krishnaswamy ,encouraged and supervised the findings of this work. All authors discussed the results and contributed to the final manuscript.

Acknowledgment

GO

None declared.

References


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